Pitofenone

Pitofenone
Names
Preferred IUPAC name
Methyl 2-{4-[2-(piperidin-1-yl)ethoxy]benzoyl}benzoate
Identifiers
CAS Number
  • 54063-52-4 checkY
3D model (JSmol)
  • Interactive image
ChemSpider
  • 108096 ☒N
PubChem CID
  • 121098
UNII
  • M09N8K7YJY checkY
CompTox Dashboard (EPA)
  • DTXSID6048381 Edit this at Wikidata
InChI
  • InChI=1S/C22H25NO4/c1-26-22(25)20-8-4-3-7-19(20)21(24)17-9-11-18(12-10-17)27-16-15-23-13-5-2-6-14-23/h3-4,7-12H,2,5-6,13-16H2,1H3 ☒N
    Key: NZHMAQSCHUSSSJ-UHFFFAOYSA-Nanalgesics ☒N
  • InChI=1/C22H25NO4/c1-26-22(25)20-8-4-3-7-19(20)21(24)17-9-11-18(12-10-17)27-16-15-23-13-5-2-6-14-23/h3-4,7-12H,2,5-6,13-16H2,1H3
    Key: NZHMAQSCHUSSSJ-UHFFFAOYAG
  • COC(=O)C1=CC=CC=C1C(=O)C2=CC=C(C=C2)OCCN3CCCCC3
Properties
Chemical formula
 C22H25NO4
Molar mass 367.445 g·mol−1
Melting point 168-169 °C (Hydrochloride)[1]
Pharmacology
A03DA02 (WHO)
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
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Infobox references
Chemical compound

Pitofenone is an antispasmodic.

Pitofenone is typically used in combination with fenpiverinium bromide, and metamizole sodium. Previously produced as Baralgin by Sanofi Aventis, the drug is currently sold in Eastern Europe under various trade names, including Spasmalgon (Actavis, Bulgaria), Revalgin (Shreya, India), Spasgan (Wockhardt, India), Bral (Micro Labs, India), and others.[2] It relieves pain and spasms of smooth muscles.[3]

References

  1. ^ Entry on Pitofenon. at: Römpp Online. Georg Thieme Verlag, retrieved 22. Juni 2019.
  2. ^ "Fenpiverinium/Metamizole/Pitofenone generic. Price of fenpiverinium/Metamizole/Pitofenone. Uses, Dosage, Side effects".
  3. ^ "Спазмалгон (Spasmalgon) - цена, листовка | Лекарства | MEDICINE.BG ®".


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