ATC代码 (L02)

ATC代码
L 抗肿瘤药及免疫制剂(Antineoplastic and immunomodulating agents)
L01 抗肿瘤药(Antineoplastic agents)
L02 内分泌治疗(Endocrine therapy)
L03 免疫增强剂(Immunostimulants)
L04 免疫抑制剂(Immunosuppressants)

A·B·C·D·G·H·QI·J·L·M·N·P·R·S·V

ATC代码L02(内分泌疗法)是解剖学治疗学及化学分类系统的一个药物分组,这是由世界卫生组织药物统计方法整合中心(The WHO Collaborating Centre for Drug Statistics Methodology)所制定的药品及其它医用产品的官方分类系统。分组L02是L抗肿瘤药及免疫用药的一部分。[1]

兽用代码(ATCvet码)可以在人用ATC代码前加Q字母:QL02[2]

国家ATC分类可能包括列表中没有的其它分类,列表为世界卫生组织(WHO)版本。

L02AA 雌激素类(Estrogens)

L02AA01 己烯雌酚(Diethylstilbestrol)
L02AA02 聚雌二醇磷酸酯(Polyestradiol phosphate)
L02AA03 炔雌醇(Ethinylestradiol)
L02AA04 磷雌酚(Fosfestrol)

L02AB 孕激素类(Progestogens)

L02AB01 甲地孕酮(Megestrol)
L02AB02 甲羟孕酮(Medroxyprogesterone)
L02AB03 孕诺酮(Gestonorone)

L02AE 促性腺素释放激素同系物(Gonadotropin-releasing hormone analogues)

L02AE01 布舍瑞林(Buserelin)
L02AE02 亮丙瑞林(Leuprorelin)
L02AE03 戈舍瑞林(Goserelin)
L02AE04 曲普瑞林(Triptorelin)

L02AX 其它激素(Other hormones)

L02BA 抗雌激素类(Anti-estrogens)

L02BA01 他莫昔芬(Tamoxifen)
L02BA02 托瑞米芬(Toremifene)
L02BA03 氟维司群(Fulvestrant)

L02BB 抗雄激素类(Anti-androgens)

L02BB01 氟他胺(Flutamide)
L02BB02 尼鲁米特(Nilutamide)
L02BB03 比卡鲁胺(Bicalutamide)

L02BG 酶抑制药类(Aromatase inhibitors)

L02BG01 氨鲁米特(Aminogluthetimide)
L02BG02 福美坦(Formestane)
L02BG03 阿那曲唑(Anastrozole)
L02BG04 来曲唑(Letrozole)
L02BG05 伏氯唑(Vorozole)
L02BG06 依西美坦(Exemestane)
L02BX01 阿巴瑞克(Abarelix)
L02BX02 地格瑞克(Degarelix)
L02BX03 阿比特龙(Abiraterone)


参考文献

  1. ^ ATC Index. WHO Collaborating Centre for Drug Statistics Methodology. 
  2. ^ ATCvet Index. WHO Collaborating Centre for Drug Statistics Methodology. 


受体
AR (A, B)


注意:此处包括了那些只有微弱男性化效应(或抗男性化(如氧雄龙))的蛋白同化甾类(因为它们合成代谢效应也是通过激活雄激素受体而是显得)。

  • Mixed (SARMs): AC-262,356
  • Andarine
  • BMS-564,929
  • Enobosarm
  • LGD-2226
  • LGD-3303
  • S-23
  • S-40503

(抑制剂)
  • 22-ABC
  • 3,3′-Dimethoxybenzidine
  • 3-Methoxybenzidine
  • Aminoglutethimide
  • Cyanoketone
  • Danazol
  • Etomidate
  • Mitotane
  • Trilostane
17α-羟化酶,
17,20-裂合酶
3β-HSD (I, II)
17β-HSD (I-XIV)
  • Danazol
  • Simvastatin
5α還原酶 (I, II)
  • 22-Oxime
  • Alfatradiol
  • Azelaic acid
  • β-Sitosterol
  • Bexlosteride
  • Dutasteride
  • 表睾酮
  • Epristeride
  • Finasteride
  • Izonsteride
  • L-39
  • Lapisteride
  • Polyunsaturated fatty acids (α-linolenic acid, linoleic acid, γ-linolenic acid, oleic acid)
  • Turosteride
  • Vitamin B6
  • 1,4,6-Androstatriene-3,17-dione
  • 4-Androstene-3,6,17-trione
  • 4-Cyclohexylaniline
  • 4-Hydroxytestosterone
  • 5α-DHNET
  • Abyssinone II
  • Aminoglutethimide
  • Anastrozole
  • 抗坏血酸维生素C
  • Atamestane
  • Bifonazole
  • CGP-45,688
  • CGS-47,645
  • Clotrimazole
  • 双氢睾酮
  • Difeconazole
  • Econazole
  • Exemestane
  • Fadrozole
  • Fenarimol
  • Finrozole
  • Formestane
  • Imazalil
  • Isoconazole
  • Ketoconazole
  • Letrozole
  • Liarozole
  • MEN-11066
  • Miconazole
  • Minamestane
  • Nimorazole
  • NKS01
  • ORG-33,201
  • Penconazole
  • Plomestane
  • Prochloraz
  • Propioconazole
  • Pyridoglutethimide
  • Rogletimide
  • Rotenone
  • Talarozole
  • Testolactone
  • Tioconazole
  • Triadimefon
  • Triadimenol
  • Troglitazone
  • Vorozole
  • YM511

Note: 21-Hydroxylase inhibitors may also affect androgen levels as they prevent metabolism of androgen steroid precursors.

其他
间接
  • Estrogens/Antiestrogens (see here)
  • GnRH agonists/antagonists (see here)
  • Gonadotropins/Antigonadotropins (see here)
  • Plasma proteins (SHBG, ABP, Albumin)
  • Progestogens/Antiprogestins (see here)
  • Prolactin
雌激素受体英语Estrogen receptor调节剂
受体
雌激素受体 (雌激素受体α, 雌激素受体β)
  • 激动剂: 3β-雄烷二醇
  • 16α-羟基雌酮
  • Alestramustine英语Alestramustine
  • Almestrone
  • 苯雌酚
  • Bifluranol英语Bifluranol
  • Broparestrol英语Broparestrol
  • Carbestrol英语Carbestrol
  • Chlorotrianisene英语Chlorotrianisene
  • Cloxestradiol英语Cloxestradiol
  • 大豆苷元
  • DHEA
  • 己二烯雌酚
  • 己烯雌酚
  • 己烯雌酚二磷酸酯
  • 薯蓣皂苷配基
  • Doisynoestrol英语Doisynoestrol
  • DPN英语Diarylpropionitrile
  • Epiestriol英语Epiestriol
  • 表美雌醇
  • Eptamestrol英语Eptamestrol/Etamestrol
  • ERB-041
  • 马萘雌酮
  • 马烯雌酮
  • 雌四醇
  • 雌二醇
  • (雌二醇苯甲酸酯
  • Estradiol butyrylacetate英语Estradiol butyrylacetate
  • Estradiol cypionate英语Estradiol cypionate
  • Estradiol dienanthate英语Estradiol dienanthate
  • Estradiol dipropionate英语Estradiol dipropionate
  • Estradiol diundecylate英语Estradiol diundecylate
  • Estradiol diundecylenate英语Estradiol diundecylenate
  • Estradiol enanthate英语Estradiol enanthate
  • Estradiol furoate英语Estradiol furoate
  • Estradiol hemisuccinate
  • Estradiol hexahydrobenzoate英语Estradiol hexahydrobenzoate
  • Estradiol monopropionate英语Estradiol monopropionate
  • Estradiol palmitate英语Estradiol palmitate
  • Estradiol pivalate英语Estradiol pivalate
  • Estradiol propoxyphenylpropionate英语Estradiol propoxyphenylpropionate
  • Estradiol stearate英语Estradiol stearate
  • Estradiol succinate英语Estradiol succinate
  • Estradiol undecylate英语Estradiol undecylate
  • 雌二醇戊酸酯)
  • Estramustine英语Estramustine
  • Estramustine phosphate英语Estramustine phosphate
  • Estrapronicate英语Estrapronicate
  • Estrazinol英语Estrazinol
  • 雌三醇
  • Estriol succinate英语Estriol succinate
  • Estriol tripropionate英语Estriol tripropionate
  • Estrofurate英语Estrofurate
  • Estromustine英语Estromustine
  • 雌酮
  • Estrone acetate英语Estrone acetate
  • Estrone cyanate英语Estrone cyanate
  • 硫酸雌酮
  • Estrone tetraacetylglucoside英语Estrone tetraacetylglucoside
  • Estropipate英语Estropipate
  • Etamestrol
  • 炔雌醇
  • Ethinylestradiol 3-isopropylsulfonate
  • Etynodiol diacetate英语Etynodiol diacetate
  • FERb 033
  • Fenestrel英语Fenestrel
  • Fosfestrol英语Fosfestrol
  • Furostilbestrol英语Furostilbestrol
  • 己烷雌酚
  • 己烷雌酚二醋酸酯
  • Hexestrol dicaprylate英语Hexestrol dicaprylate
  • Hexestrol diphosphate英语Hexestrol diphosphate
  • Hexestrol dipropionate英语Hexestrol dipropionate
  • Hydroxyestrone diacetate英语Hydroxyestrone diacetate
  • Liquiritigenin英语Liquiritigenin
  • 美雌醇
  • Methallenestril英语Methallenestril
  • Methestrol
  • Methestrol dipropionate英语Methestrol dipropionate
  • 莫克雌醇
  • Nilestriol英语Nilestriol
  • Orestrate英语Orestrate
  • 聚磷酸雌二醇
  • PPT
  • Promestriene英语Promestriene
  • Promethoestrol英语Promethoestrol
  • Quinestradol英语Quinestradol
  • Quinestrol英语Quinestrol
  • Β-穀固醇
  • WAY-200,070

Note: Though not listed here, many anabolic steroids can also be estrogenic as they can be aromatized into estrogen-like metabolites that possess estrogenic activity.

  • 混合(選擇性雌激素受體調節物):2-羥基雌酮
  • 醋氟拉诺
  • 阿考比芬英语Acolbifene
  • 阿非昔芬英语Afimoxifene
  • 双炔失碳醇
  • 双炔失碳酯
  • 阿佐昔芬英语Arzoxifene
  • 巴多昔芬英语Bazedoxifene
  • 布林司群
  • 溴帕雌烯
  • 卡米司群
  • 氯烯雌醚
  • 氯米芬
  • 氧氯米芬英语Clomifenoxide
  • CN-55945-27
  • 环芬尼英语Cyclofenil
  • D-15413
  • 去甲基氯烯雌醚
  • 屈洛昔芬英语Droloxifene
  • 恩氯米芬英语Enclomifene
  • 内昔芬
  • 表美雌醇
  • 依他舒
  • 乙胺氧三苯醇
  • Femarelle英语Femarelle
  • 非培米芬英语Fispemifene
  • GW5638
  • ICI-55548
  • 艾多昔芬英语Idoxifene
  • 拉索昔芬英语Lasofoxifene
  • 左美洛昔芬英语Levormeloxifene
  • LN-1643
  • LN-2299
  • LY-117018
  • Menerba英语Menerba
  • 美雄烷英语Mepitiostane
  • 米泼昔芬英语Miproxifene
  • 磷酸米泼昔芬
  • MRL-37
  • 萘福昔定英语Nafoxidine
  • 硝米芬英语Nitromifene
  • NNC 45-0095
  • NNC 45-0320
  • NNC 45-0781
  • NNC 45-1506
  • 奥美昔芬英语Ormeloxifene
  • 奥培米芬英语Ospemifene
  • 帕诺米芬
  • 哌喷昔芬英语Pipendoxifene
  • 普林贝瑞英语Prinaberel
  • 雷洛昔芬
  • SS1010
  • 司韦芬英语Sivifene
  • 他莫昔芬
  • TAS-108
  • 替米利芬英语Tesmilifene
  • 替勃龙英语Tibolone
  • 托瑞米芬
  • 曲沃昔芬英语Trioxifene
  • TZE-5323
  • U-11555A
  • U-11634
  • Y-134
  • 秦哚昔芬
  • 珠氯米芬英语Zuclomifene
  • 拮抗剂:
  • Fulvestrant英语Fulvestrant
  • ICI-164,384
  • MPP
  • PHTPP
  • RU-58,668
  • SS1020
  • ZK-164,015
  • ZK-191,703

脚注: 不包括環境雌激素(例如植物雌激素和黴菌雌激素)。完整環境雌激素見此英语Template:Xenoestrogens

G蛋白偶联雌激素受体
  • 拮抗剂: G-15

(抑制剂)
  • 22-ABC
  • 3,3′-Dimethoxybenzidine
  • 3-Methoxybenzidine
  • Aminoglutethimide英语Aminoglutethimide
  • Cyanoketone英语Cyanoketone
  • 達那唑
  • Etomidate英语Etomidate
  • Mitotane英语Mitotane
  • Trilostane英语Trilostane
17α-羟基化酶
17,20-碳链裂解酶
3β-HSD英语3β-Hydroxysteroid dehydrogenase
  • 1,4,6-Androstatriene-3,17-dione英语1,4,6-Androstatriene-3,17-dione
  • 4-雄烯-3,6,17-三酮
  • 4-Cyclohexylaniline
  • 4-Hydroxytestosterone英语4-Hydroxytestosterone
  • 5α-DHNET英语5α-Dihydro-19-norethisterone
  • Abyssinone II
  • Aminoglutethimide英语Aminoglutethimide
  • Anastrozole英语Anastrozole
  • 抗壞血酸維生素C
  • Atamestane英语Atamestane
  • 聯苯芐唑
  • CGP-45,688
  • CGS-47,645
  • 克催瑪汝
  • DHT
  • Difeconazole
  • 益康唑
  • 依西美坦
  • Fadrozole英语Fadrozole
  • Fenarimol英语Fenarimol
  • Finrozole英语Finrozole
  • Formestane英语Formestane
  • 抑霉唑
  • Isoconazole英语Isoconazole
  • 酮康唑
  • 來曲唑
  • Liarozole英语Liarozole
  • MEN-11066
  • 咪康唑
  • Minamestane英语Minamestane
  • Nimorazole英语Nimorazole
  • NKS01
  • ORG-33,201
  • 戊菌唑
  • 普洛美坦
  • 咪鲜胺
  • 丙环唑
  • Pyridoglutethimide英语Pyridoglutethimide
  • Rogletimide
  • 魚藤酮
  • Talarozole英语Talarozole
  • Testolactone英语Testolactone
  • 噻康唑
  • Triadimefon英语Triadimefon
  • 三唑醇
  • Troglitazone英语Troglitazone
  • Vorozole英语Vorozole
  • YM511

Note: 5α-reductase and 21-hydroxylase英语21-hydroxylase inhibitors may also affect estrogen levels as they prevent metabolism of estrogen steroid precursors.

Other
Indirect
孕酮受体調控劑英语receptor modulator
PR
受體致活劑
  • 3,8-Dihydrodiligustilide
  • 5α-Dihydroprogesterone英语5α-Dihydroprogesterone
  • 6,6-Difluoronorethisterone
  • 7α-Methylmetribolone (7α,17α-dimethyltrenbolone)英语7α-Methylmetribolone
  • 9α-Bromo-11-ketoprogesterone
  • 11β-Methyl-19-nortestosterone
  • 11β-Methyl-19-nortestosterone 17β-dodecylcarbonate
  • 11-Dehydroprogesterone
  • 11-脱氧皮质酮
  • 17α-Hydroxyprogesterone英语17α-Hydroxyprogesterone
  • 17α-Methylprogesterone英语17α-Methylprogesterone
  • 19-Norprogesterone英语19-Norprogesterone
  • 20α-Dihydroprogesterone英语20α-Dihydroprogesterone
  • Δ4-Tibolone
  • Acetomepregenol (mepregenol diacetate)英语Acetomepregenol
  • Algestone英语Algestone
  • Algestone acetonide英语Algestone acetonide
  • Algestone acetophenide英语Algestone acetophenide
  • Allylestrenol英语Allylestrenol
  • Altrenogest英语Altrenogest
  • Amadinone英语Amadinone
  • Amadinone acetate英语Amadinone acetate
  • Anagestone英语Anagestone
  • Anagestone acetate英语Anagestone acetate
  • Bolandiol英语Bolandiol
  • Bolandiol dipropionate英语Bolandiol dipropionate
  • Butagest
  • Buterol
  • Canrenoic acid英语Canrenoic acid
  • Canrenone英语Canrenone
  • Chlormadinone英语Chlormadinone
  • Chlormadinone acetate英语Chlormadinone acetate
  • Chloroethynyl norgestrel英语Chloroethynyl norgestrel
  • Cingestol英语Cingestol
  • Cismadinone英语Cismadinone
  • Cismadinone acetate英语Cismadinone acetate
  • Clogestone英语Clogestone
  • Clogestone acetate英语Clogestone acetate
  • Clomegestone英语Clomegestone
  • Clomegestone acetate英语Clomegestone acetate
  • 醋酸环丙孕酮
  • Danazol英语Danazol
  • Delmadinone英语Delmadinone
  • Delmadinone acetate英语Delmadinone acetate
  • Demegestone英语Demegestone
  • Desogestrel英语Desogestrel
  • Dienogest英语Dienogest
  • 二甲孕烯
  • Dimethandrolone英语Dimethandrolone
  • Dimethandrolone undecanoate
  • Dimethisterone英语Dimethisterone
  • 薯蓣皂苷配基
  • Drospirenone英语Drospirenone
  • Dydrogesterone英语Dydrogesterone
  • Edogestrone英语Edogestrone
  • Ethisterone英语Ethisterone
  • Ethynerone英语Ethynerone
  • Etonogestrel英语Etonogestrel
  • Etynodiol英语Etynodiol
  • Etynodiol diacetate英语Etynodiol diacetate
  • Flugestone英语Flugestone
  • 醋酸氟孕酮
  • Gestaclone英语Gestaclone
  • Gestadienol英语Gestadienol
  • Gestodene英语Gestodene
  • Gestonorone caproate (gestronoly hexanoate)英语Gestonorone caproate
  • Gestrinone英语Gestrinone
  • Gestronol (gestonorone)英语Gestronol
  • Haloprogesterone英语Haloprogesterone
  • Hydromadinone英语Hydromadinone
  • Hydroxyprogesterone acetate英语Hydroxyprogesterone acetate
  • Hydroxyprogesterone butyrate
  • Hydroxyprogesterone caproate (hydroxyprogesterone hexanoate)英语Hydroxyprogesterone caproate
  • Hydroxyprogesterone heptanoate (hydroxyprogesterone enanthate)英语Hydroxyprogesterone heptanoate
  • 左炔诺孕酮
  • Lynestrenol英语Lynestrenol
  • Mecigestone (pentarane B)
  • Medrogestone英语Medrogestone
  • Medroxyprogesterone英语Medroxyprogesterone
  • Medroxyprogesterone acetate英语Medroxyprogesterone acetate
  • Megestrol英语Megestrol
  • Megestrol acetate英语Megestrol acetate
  • Melengestrol英语Melengestrol
  • Melengestrol acetate英语Melengestrol acetate
  • Mespirenone英语Mespirenone
  • Methylestrenolone英语Methylestrenolone
  • Metribolone (R1881)英语Metribolone
  • Metynodiol英语Metynodiol
  • Metynodiol diacetate英语Metynodiol diacetate
  • Methoxydienone (methoxygonadiene)
  • Mometasone furoate英语Mometasone furoate
  • Nandrolone英语Nandrolone
  • Nandrolone ester英语Nandrolone esters (e.g., nandrolone phenylpropionate英语nandrolone phenylpropionate, nandrolone decanoate英语nandrolone decanoate)
  • Nomegestrol英语Nomegestrol
  • Nomegestrol acetate英语Nomegestrol acetate
  • Norelgestromin英语Norelgestromin
  • Norethisterone (norethindrone)英语Norethisterone
  • Norethisterone acetate英语Norethisterone acetate
  • Norethisterone acetate oxime英语Norethisterone acetate oxime
  • Norethisterone enanthate英语Norethisterone enanthate
  • Noretynodrel英语Noretynodrel
  • Norgesterone英语Norgesterone
  • Norgestimate英语Norgestimate
  • Norgestomet英语Norgestomet
  • Norgestrel英语Norgestrel
  • Norgestrienone英语Norgestrienone
  • Norvinisterone英语Norvinisterone
  • ORG-2058
  • Osaterone英语Osaterone
  • Osaterone acetate英语Osaterone acetate
  • Oxendolone英语Oxendolone
  • Oxogestone英语Oxogestone
  • Oxogestone phenpropionate英语Oxogestone phenpropionate
  • Pentagestrone英语Pentagestrone
  • Pentagestrone acetate英语Pentagestrone acetate
  • Pentarane A
  • Potassium canrenoate英语Potassium canrenoate
  • 孕酮
  • Proligestone英语Proligestone
  • Promegestone英语Promegestone
  • Quingestanol英语Quingestanol
  • Quingestanol acetate英语Quingestanol acetate
  • Retroprogesterone英语Retroprogesterone
  • Ro 6-3129
  • Riligustilide
  • SC-5233英语SC-5233
  • SC-8109
  • Segesterone英语Segesterone
  • Segesterone acetate (nestorone)英语Nestorone
  • 螺内酯
  • Spirorenone英语Spirorenone
  • Tanaproget英语Tanaproget
  • Tetrahydrogestrinone英语Tetrahydrogestrinone
  • Tibolone英语Tibolone
  • Tigestol英语Tigestol
  • Tosagestin英语Tosagestin
  • Trengestone英语Trengestone
  • Trestolone英语Trestolone
  • Trestolone acetate英语Trestolone acetate
  • Trimegestone英语Trimegestone
  • ZM-182345
Mixed (SPRMs英语Selective progesterone receptor modulator)
  • Apigenin英语Apigenin
  • Asoprisnil英语Asoprisnil
  • Asoprisnil ecamate
  • Guggulsterone英语Guggulsterone
  • 山柰酚
  • J1042
  • LG-120838
  • Naringenin英语Naringenin
  • PRA-910
  • 丁香酸
  • Telapristone英语Telapristone
  • 受體拮抗劑: 美服培酮
  • Org-31710
  • Org-33628
  • Ulipristal acetate英语Ulipristal acetate
  • ZK-137316
Antagonists
mPRs英语Membrane progesterone receptor
(PAQRs英语Progestin and adipoQ receptor)
受體致活劑
  • 5α-Dihydroprogesterone英语5α-Dihydroprogesterone
  • 5β-Dihydroprogesterone英语5β-Dihydroprogesterone
  • 11-脱氧皮质酮
  • 17α-Hydroxyprogesterone英语17α-Hydroxyprogesterone
  • 17α,21-Dihydroxyprogesterone
  • Allopregnanolone英语Allopregnanolone
  • 美服培酮
  • 孕烯醇酮
  • 孕酮
Antagonists
參見: 雄激素 • 雌激素 • Glucocorticoidics • Mineralocorticoidics